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Table 2 Examples of exceptions to midazolam classification for seven CYP3A4 inhibitors

From: A useful tool for drug interaction evaluation: The University of Washington Metabolism and Transport Drug Interaction Database

Inhibitor Classification with sensitive substrate Sensitive substrate
Potent with midazolam
Clarithromycin moderate saquinavir
Ketoconazole moderate saquinavir
Nefazodone moderate triazolam
Troleandomycin moderate triazolam
Moderate with midazolam
Erythromycin potent simvastatin/buspirone
Diltiazem potent buspirone
Fluconazole weak saquinavir